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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T10248 | Adenosine antagonist-1 | Adenosine Receptor | |
Adenosine antagonist-1 acts as an adenosine A3 receptor (AA3R) antagonist. | |||
T40307 | Adenosine receptor antagonist 1 | ||
Adenosine receptor antagonist 1 is a highly selective antagonist for the A2aR adenosine receptor, exhibiting an IC50 value of 0.29 nM. It demonstrates a remarkable 14-fold selectivity towards the A2aR receptor in compari... | |||
T37792 | A2A receptor antagonist 1 | CPI-444 analog,A2A receptor antagonist 1 | Adenosine Receptor |
A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively. | |||
T10058 | A2B receptor antagonist 1 | Adenosine Receptor | |
A2B receptor antagonist 1 (EXAMPLE 9B) is a potent A2B adenosine receptor antagonist. | |||
T8312 | Derenofylline | Adenosine Receptor | |
Derenofylline is a selective and potent adenosine A(1) antagonist in vitro (Ki=1 nM) | |||
T15418 | GS-6201 | CVT-6883 | Adenosine Receptor |
GS-6201 (CVT-6883) is a selective antagonist of adenosine A2B receptor. GS-6201 shows high affinity and selectivity for the human adenosine A2B receptors with a Ki of 22 nM. | |||
T14078 | AB928 | Adenosine Receptor | |
AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1]. | |||
T22031 | ANR 94 | Adenosine Receptor | |
ANR94 is a potent, selective antagonist of the adenosine A2A receptor (AA2AR), exhibiting a K_i value of 46 nM for the human AA2AR (hAA2AR). This compound shows promise for research into Parkinson's disease. [1] [2] | |||
T70648 | FK-352 | ||
FK-352 is a pyrazolopyridine derivative and adenosine-1 receptor antagonist. | |||
T24384 | L-97-1 | L97-1,L 97-1 | |
L-97-1 is an antagonist of the adenosine A1 receptor. | |||
T62611 | Adenosine receptor antagonist 2 | ||
Adenosine receptor antagonist 2 is an orally active A2a (IC50: 1 nM), A2b (IC50: 3 nM) adenosine receptor antagonist that exhibits antitumour effects. | |||
T70996 | FK-838 | ||
FK-838 is an adenosine subtype-1 receptor antagonist. | |||
T60872 | Adenosine receptor antagonist 3 | ||
Adenosine receptor antagonist 3 has the potential for cancer disease research which is a potent adenosine receptor antagonist [1]. | |||
T72000 | N 0840 | ||
N 0840 is a selective, orally active A(1) adenosine receptor antagonist. | |||
T61850 | Adenosine receptor inhibitor 1 | ||
Adenosine receptor inhibitor 1 is a highly potent and selective antagonist of adenosine receptor (AR). It exhibits exceptional affinity for A1 AR, A2A AR, A2B AR, and A3 AR, with respective Ki values of >1000, 68.5, >100... | |||
T60580 | A1AR antagonist 2 | ||
A1AR antagonist 2 (compound 18h) is a potent antagonist of the A1 adenosine receptor (AR). A1AR antagonist 2 has Ki values of 1.49, 10.2, and 50.1 nM for hA 1, hA 2A, and hA 2B, respectively [1]. | |||
T62134 | A1/A3 AR antagonist 1 | ||
A1/A3 AR antagonist 1 (Compound 10) is a potent, dual adenosine 1 (A1) and adenosine 3 (A3) receptor antagonist that acts on human A1 (Ki: 37.6 nM), human A3 (Ki: 25.4 nM) and rat A1 (Ki: 1.47 nM). 1 Can be used to study... | |||
T61536 | A1AR antagonist 4 | ||
A1AR antagonist 4 (compound 22) is a highly developed chemical compound that acts as a potent and selective antagonist of the A1 adenosine receptor (A1AR). It possesses a pIC50 value of 5.51 and a pKi value of 6.29 [1]. | |||
T60687 | A1AR antagonist 1 | ||
A1AR antagonist 1 (compound 18g) is a potent antagonist of A1 adenosine receptor (AR). A1AR antagonist 1 has Ki values of 2.08, 6.91, and 31.2 nM for hA1, hA2A and hA2B, respectively [1]. | |||
T60615 | A1AR antagonist 6 | ||
A1AR antagonist 6 (compound 15) is a potent and selective antagonist of A1 adenosine receptor(A1AR) with a pKi of 7.13 and a pIC 50 of 6.38[1]. |